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rdf:type |
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lifeskim:mentions |
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pubmed:issue |
7
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pubmed:dateCreated |
2010-3-22
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pubmed:abstractText |
The identification of novel, potent, non-steroidal/small molecule functional GR antagonist GSK1564023A selective over PR is described. Associated structure-activity relationships and the process of optimisation of an initial HTS hit are also described.
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pubmed:language |
eng
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pubmed:journal |
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pubmed:citationSubset |
IM
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pubmed:chemical |
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pubmed:status |
MEDLINE
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pubmed:month |
Apr
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pubmed:issn |
1464-3405
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pubmed:author |
pubmed-author:BerthelemeNicolasN,
pubmed-author:BrownDavidD,
pubmed-author:CairnsWilliamW,
pubmed-author:CaivanoMatildeM,
pubmed-author:D'AlessandroPierP,
pubmed-author:DunneAngelaA,
pubmed-author:GrayDavidD,
pubmed-author:GulSherazS,
pubmed-author:HunjanSuchete SSS,
pubmed-author:MontanariDinoD,
pubmed-author:RimlandJosephJ,
pubmed-author:SasseRosemaryR,
pubmed-author:ShahPoonamP,
pubmed-author:SmithDavid NDN,
pubmed-author:SmithPaul WPW,
pubmed-author:StandingDavidD,
pubmed-author:TrumpRyanR,
pubmed-author:UingsIainI,
pubmed-author:VimalMythilyM,
pubmed-author:WatsonStephen PSP
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pubmed:copyrightInfo |
2010 Elsevier Ltd. All rights reserved.
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pubmed:issnType |
Electronic
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pubmed:day |
1
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pubmed:volume |
20
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pubmed:owner |
NLM
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|
pubmed:authorsComplete |
Y
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pubmed:pagination |
2340-3
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pubmed:meshHeading |
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pubmed:year |
2010
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pubmed:articleTitle |
The identification a novel, selective, non-steroidal, functional glucocorticoid receptor antagonist.
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pubmed:affiliation |
Medicines Research Centre, Verona, Italy.
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pubmed:publicationType |
Journal Article
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