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pubmed-article:9990463pubmed:abstractTextNovel 2,6,9-substituted purine derivatives represent a class of potent and selective inhibitors of CDK1/cyclinB. The synthesis, SAR and biological profile of selected compounds are described.lld:pubmed
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pubmed-article:9990463pubmed:articleTitle2,6,9-trisubstituted purines: optimization towards highly potent and selective CDK1 inhibitors.lld:pubmed
pubmed-article:9990463pubmed:affiliationNovartis Pharmaceuticals, Novartis Limited, Basel, Switzerland.lld:pubmed
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