pubmed:abstractText |
The syntheses of 11-ethyl and 11-cyclopropyldipyrido[2,3-b:3',2'-f]azepines, analogs of the HIV-1 reverse transcriptase inhibitor nevirapine 1, are described. These compounds exhibit potency equivalent to nevirapine in the inhibition of wild-type and some mutant RT enzymes.
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pubmed:affiliation |
Department of Chemical Development, Boehringer Ingelheim Pharmaceuticals, Inc., Ridgefield, CT 06877, USA.
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