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pubmed-article:8622120pubmed:abstractTextWe developed new biochemical approaches to demonstrate the presence of inositol 1,4,5-triphosphate (InsP3)-gated calcium channels in presynaptic plasma membranes (SPM) and their involvement in the presynaptic receptor-mediated Ca2+ influx into nerve terminals. In perfusion experiments using SPM vesicles preloaded with 45Ca2+, InsP3 elicited the release of 45CA2+ into perfusates in a saturable manner. The InsP3- evoked 45Ca2+ release from resealed SPM vesicles was more potent than that from resealed vesicles using any other subcellular fractions. Here we also report the involvement of InsP3-gated mechanisms in the presynaptic receptor-mediated Ca2+ influx into synaptosomes (nerve terminals) by use of such resealed vesicles reconstituted with purified Gi1.lld:pubmed
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pubmed-article:8622120pubmed:articleTitleInositol 1,4,5-trisphosphate-gated calcium transport through plasma membranes in nerve terminals.lld:pubmed
pubmed-article:8622120pubmed:affiliationDepartment of Pharmacology, Yokohama City University School of Medicine, Japan.lld:pubmed
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