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pubmed-article:19362479pubmed:abstractTextA series of trifluoromethyl, benzothiazolyl or thiazolyl ketone-containing peptidic compounds as SARS-CoV 3CL protease inhibitors were developed and their potency was evaluated by in vitro protease inhibitory assays. Three candidates had encouraging results for the development of new anti-SARS compounds.lld:pubmed
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pubmed-article:19362479pubmed:articleTitleNew developments for the design, synthesis and biological evaluation of potent SARS-CoV 3CL(pro) inhibitors.lld:pubmed
pubmed-article:19362479pubmed:affiliationDepartment of Medicinal Chemistry, Center for Frontier Research in Medicinal Science, Kyoto Pharmaceutical University, Japan.lld:pubmed
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