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18482836
Source:
http://linkedlifedata.com/resource/pubmed/id/18482836
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rdf:type
pubmed:Citation
lifeskim:mentions
umls-concept:C0031809
,
umls-concept:C0034251
,
umls-concept:C0243077
,
umls-concept:C1167622
pubmed:issue
11
pubmed:dateCreated
2008-5-30
pubmed:abstractText
A potent IRAK-4 inhibitor was identified through routine project cross screening. The binding mode was inferred using a combination of in silico docking into an IRAK-4 homology model, surrogate crystal structure analysis and chemical analogue SAR.
pubmed:language
eng
pubmed:journal
http://linkedlifedata.com/resource/pubmed/journal/9107377
pubmed:citationSubset
IM
pubmed:chemical
http://linkedlifedata.com/resource/pubmed/chemical/Enzyme Inhibitors
,
http://linkedlifedata.com/resource/pubmed/chemical/Imidazoles
,
http://linkedlifedata.com/resource/pubmed/chemical/Interleukin-1 Receptor-Associated...
,
http://linkedlifedata.com/resource/pubmed/chemical/Pyridines
pubmed:status
MEDLINE
pubmed:month
Jun
pubmed:issn
1464-3405
pubmed:author
pubmed-author:BuckleyGeorge MGM
,
pubmed-author:CeskaThomas ATA
,
pubmed-author:FraserJoanne LJL
,
pubmed-author:GowersLewisL
,
pubmed-author:GroomColin RCR
,
pubmed-author:HiguerueloAlicia PerezAP
,
pubmed-author:JenkinsKerryK
,
pubmed-author:MackStephen RSR
,
pubmed-author:MorganTrevorT
,
pubmed-author:ParryDavid MDM
,
pubmed-author:PittWilliam RWR
,
pubmed-author:RauschOliverO
,
pubmed-author:RichardMarianna DMD
,
pubmed-author:SabinVerityV
pubmed:issnType
Electronic
pubmed:day
1
pubmed:volume
18
pubmed:owner
NLM
pubmed:authorsComplete
Y
pubmed:pagination
3291-5
pubmed:dateRevised
2009-11-19
pubmed:meshHeading
pubmed-meshheading:18482836-Binding Sites
,
pubmed-meshheading:18482836-Crystallography, X-Ray
,
pubmed-meshheading:18482836-Drug Design
,
pubmed-meshheading:18482836-Enzyme Inhibitors
,
pubmed-meshheading:18482836-Imidazoles
,
pubmed-meshheading:18482836-Interleukin-1 Receptor-Associated Kinases
,
pubmed-meshheading:18482836-Models, Molecular
,
pubmed-meshheading:18482836-Molecular Conformation
,
pubmed-meshheading:18482836-Molecular Structure
,
pubmed-meshheading:18482836-Pyridines
,
pubmed-meshheading:18482836-Structure-Activity Relationship
pubmed:year
2008
pubmed:articleTitle
IRAK-4 inhibitors. Part II: a structure-based assessment of imidazo[1,2-a]pyridine binding.
pubmed:affiliation
UCB, Granta Park, Great Abington, Cambridge CB21 6GS, UK.
pubmed:publicationType
Journal Article