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pubmed-article:17936624pubmed:abstractTextWe describe three novel regioisomeric series of aryl naphthyridine analogs, which are potent antagonists of the Class III GPCR mGlu5 receptor. The synthesis and in vitro and in vivo pharmacological activities of these analogs are discussed.lld:pubmed
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pubmed-article:17936624pubmed:articleTitleSynthesis and SAR comparison of regioisomeric aryl naphthyridines as potent mGlu5 receptor antagonists.lld:pubmed
pubmed-article:17936624pubmed:affiliationDepartment of Medicinal Chemistry, Pfizer Global Research & Development, 2800 Plymouth Road, Ann Arbor, MI 48105, USA.lld:pubmed
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