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pubmed-article:15369383pubmed:abstractTextProteasome inhibition is a therapeutic concept of current interest in anticancer research. We report here the design, synthesis, and biological characterization of prototypes of a new class of noncovalent proteasome inhibitors showing high activity in biochemical and cellular assays.lld:pubmed
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pubmed-article:15369383pubmed:articleTitleEntry into a new class of potent proteasome inhibitors having high antiproliferative activity by structure-based design.lld:pubmed
pubmed-article:15369383pubmed:affiliationNovartis Pharma AG, Novartis Institutes for Biomedical Research, CH-4002 Basel, Switzerland.lld:pubmed
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