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12781182
Source:
http://linkedlifedata.com/resource/pubmed/id/12781182
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Predicate
Object
rdf:type
pubmed:Citation
lifeskim:mentions
umls-concept:C0002482
,
umls-concept:C0007428
,
umls-concept:C0243077
,
umls-concept:C2717970
pubmed:issue
12
pubmed:dateCreated
2003-6-3
pubmed:abstractText
Modeling, synthesis and in vitro activities of a series of arylaminoethyl amide based inhibitors of the cysteine protease cathepsin K are described.
pubmed:language
eng
pubmed:journal
http://linkedlifedata.com/resource/pubmed/journal/9107377
pubmed:citationSubset
IM
pubmed:chemical
http://linkedlifedata.com/resource/pubmed/chemical/Amides
,
http://linkedlifedata.com/resource/pubmed/chemical/Benzene Derivatives
,
http://linkedlifedata.com/resource/pubmed/chemical/CTSK protein, human
,
http://linkedlifedata.com/resource/pubmed/chemical/CTSL1 protein, human
,
http://linkedlifedata.com/resource/pubmed/chemical/Cathepsin K
,
http://linkedlifedata.com/resource/pubmed/chemical/Cathepsin L
,
http://linkedlifedata.com/resource/pubmed/chemical/Cathepsins
,
http://linkedlifedata.com/resource/pubmed/chemical/Cysteine Endopeptidases
,
http://linkedlifedata.com/resource/pubmed/chemical/Cysteine Proteinase Inhibitors
,
http://linkedlifedata.com/resource/pubmed/chemical/Recombinant Proteins
,
http://linkedlifedata.com/resource/pubmed/chemical/cathepsin S
pubmed:status
MEDLINE
pubmed:month
Jun
pubmed:issn
0960-894X
pubmed:author
pubmed-author:AltmannEvaE
,
pubmed-author:GreenJonathanJ
,
pubmed-author:Tintelnot-BlomleyMarinaM
pubmed:issnType
Print
pubmed:day
16
pubmed:volume
13
pubmed:owner
NLM
pubmed:authorsComplete
Y
pubmed:pagination
1997-2001
pubmed:dateRevised
2009-11-19
pubmed:meshHeading
pubmed-meshheading:12781182-Amides
,
pubmed-meshheading:12781182-Benzene Derivatives
,
pubmed-meshheading:12781182-Binding Sites
,
pubmed-meshheading:12781182-Cathepsin K
,
pubmed-meshheading:12781182-Cathepsin L
,
pubmed-meshheading:12781182-Cathepsins
,
pubmed-meshheading:12781182-Cysteine Endopeptidases
,
pubmed-meshheading:12781182-Cysteine Proteinase Inhibitors
,
pubmed-meshheading:12781182-Humans
,
pubmed-meshheading:12781182-Inhibitory Concentration 50
,
pubmed-meshheading:12781182-Models, Molecular
,
pubmed-meshheading:12781182-Recombinant Proteins
,
pubmed-meshheading:12781182-Structure-Activity Relationship
pubmed:year
2003
pubmed:articleTitle
Arylaminoethyl amides as inhibitors of the cysteine protease cathepsin K-investigating P1' substituents.
pubmed:affiliation
Arthritis & Bone Metabolism Therapeutic Area, Novartis Pharma AG, CH-4002, Basel, Switzerland, eva.altmann@pharma.novartis.com
pubmed:publicationType
Journal Article