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12639538
Source:
http://linkedlifedata.com/resource/pubmed/id/12639538
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rdf:type
pubmed:Citation
lifeskim:mentions
umls-concept:C0260181
,
umls-concept:C1257954
pubmed:issue
4
pubmed:dateCreated
2003-3-17
pubmed:abstractText
Pyridazinone was found to be an excellent core template for selective COX-2 inhibitors. Two potent, selective and orally active COX-2 inhibitors, which were highly efficacious in rat paw edema and rat pyresis models, have been obtained.
pubmed:language
eng
pubmed:journal
http://linkedlifedata.com/resource/pubmed/journal/9107377
pubmed:citationSubset
IM
pubmed:chemical
http://linkedlifedata.com/resource/pubmed/chemical/Cyclooxygenase 1
,
http://linkedlifedata.com/resource/pubmed/chemical/Cyclooxygenase 2
,
http://linkedlifedata.com/resource/pubmed/chemical/Cyclooxygenase 2 Inhibitors
,
http://linkedlifedata.com/resource/pubmed/chemical/Cyclooxygenase Inhibitors
,
http://linkedlifedata.com/resource/pubmed/chemical/Isoenzymes
,
http://linkedlifedata.com/resource/pubmed/chemical/Membrane Proteins
,
http://linkedlifedata.com/resource/pubmed/chemical/PTGS1 protein, human
,
http://linkedlifedata.com/resource/pubmed/chemical/PTGS2 protein, human
,
http://linkedlifedata.com/resource/pubmed/chemical/Prostaglandin-Endoperoxide Synthases
,
http://linkedlifedata.com/resource/pubmed/chemical/Ptgs1 protein, rat
,
http://linkedlifedata.com/resource/pubmed/chemical/Pyridazines
pubmed:status
MEDLINE
pubmed:month
Feb
pubmed:issn
0960-894X
pubmed:author
pubmed-author:BrideauChristineC
,
pubmed-author:ChanChi ChungCC
,
pubmed-author:CharlesonStellaS
,
pubmed-author:ClaveauDavidD
,
pubmed-author:GauthierJacques YvesJY
,
pubmed-author:GordonRobertR
,
pubmed-author:GreigGillianG
,
pubmed-author:LauCheuk KCK
,
pubmed-author:LiChun SingCS
,
pubmed-author:PrasitPetpiboonP
,
pubmed-author:RiendeauDenisD
,
pubmed-author:SavoieChantalC
,
pubmed-author:ThérienMichelM
,
pubmed-author:WongElizabethE
pubmed:issnType
Print
pubmed:day
24
pubmed:volume
13
pubmed:owner
NLM
pubmed:authorsComplete
Y
pubmed:pagination
597-600
pubmed:dateRevised
2005-11-17
pubmed:meshHeading
pubmed-meshheading:12639538-Animals
,
pubmed-meshheading:12639538-Cell Line
,
pubmed-meshheading:12639538-Cyclooxygenase 1
,
pubmed-meshheading:12639538-Cyclooxygenase 2
,
pubmed-meshheading:12639538-Cyclooxygenase 2 Inhibitors
,
pubmed-meshheading:12639538-Cyclooxygenase Inhibitors
,
pubmed-meshheading:12639538-Edema
,
pubmed-meshheading:12639538-Humans
,
pubmed-meshheading:12639538-Inhibitory Concentration 50
,
pubmed-meshheading:12639538-Isoenzymes
,
pubmed-meshheading:12639538-Membrane Proteins
,
pubmed-meshheading:12639538-Metabolic Clearance Rate
,
pubmed-meshheading:12639538-Prostaglandin-Endoperoxide Synthases
,
pubmed-meshheading:12639538-Pyridazines
,
pubmed-meshheading:12639538-Rats
,
pubmed-meshheading:12639538-Structure-Activity Relationship
pubmed:year
2003
pubmed:articleTitle
Pyridazinones as selective cyclooxygenase-2 inhibitors.
pubmed:affiliation
Merck Frosst Centre for Therapeutic Research, PO Box 1005, Pointe-Claire-Dorval, Quebec, Canada H9R 4P8. chunsing_li@merck.com
pubmed:publicationType
Journal Article