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pubmed-article:10465547pubmed:abstractTextExtensive SAR has been established in the alkoxy lactone series and this has lead to the discovery of DFP (5,5-dimethyl-3-(2-propoxy)-4-methanesulfonylphenyl)-2(5H)-furanon e), a potent COX-2 inhibitor exhibiting in vivo efficacy in all models studied.lld:pubmed
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pubmed-article:10465547pubmed:articleTitleSAR in the alkoxy lactone series: the discovery of DFP, a potent and orally active COX-2 inhibitor.lld:pubmed
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