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pubmed-article:9578182pubmed:abstractTextSaquinavir is a potent HIV protease inhibitor whose effectiveness is limited in vivo by its low bioavailability. Since saquinavir is metabolized by CYP3A4, the effect of grapefruit juice, an inhibitor of CYP3A4, was investigated on its bioavailability.lld:pubmed
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pubmed-article:9578182pubmed:articleTitleGrapefruit juice enhances the bioavailability of the HIV protease inhibitor saquinavir in man.lld:pubmed
pubmed-article:9578182pubmed:affiliationDivision of Clinical Pharmacology & Toxicology, University Hospital, Zürich, Switzerland.lld:pubmed
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