Inhibitors of acyl-CoA:cholesterol O-acyl transferase (ACAT) as hypocholesterolemic agents. 8. Incorporation of amide or amine functionalities into a series of disubstituted ureas and carbamates. Effects on ACAT inhibition in vitro and efficacy in vivo.

Source:http://linkedlifedata.com/resource/pubmed/id/8021920

J. Med. Chem. 1994 Jun 10 37 12 1810-22

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8021920