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pubmed-article:12873492pubmed:abstractTextHydroxylation of hypoxia-inducible factor, a nuclear transcription factor, is catalysed by iron and 2-oxoglutarate dependent hydroxylases. Various analogues of the 2-oxoglutarate cosubstrate were synthesised and shown to inhibit the activity of human hypoxia-inducible factor-1alpha prolyl hydroxylases in cell-free extracts.lld:pubmed
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pubmed-article:12873492pubmed:affiliationWellcome Trust Centre for Human Genetics, Roosevelt Drive, Oxford OX3 7BN, UK.lld:pubmed
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